Aurora B inhibitor 1

CAS No. 937276-52-3

Aurora B inhibitor 1( —— )

Catalog No. M33019 CAS No. 937276-52-3

Aurora B inhibitor 1 is an Aurora B (Aurora-1) inhibitor (Ki <0.010 μM) with potential anticancer activity for cancer research.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Aurora B inhibitor 1
  • Note
    Research use only, not for human use.
  • Brief Description
    Aurora B inhibitor 1 is an Aurora B (Aurora-1) inhibitor (Ki <0.010 μM) with potential anticancer activity for cancer research.
  • Description
    Aurora B inhibitor 1 is an Aurora B (Aurora-1) inhibitor extracted from patent WO2007059299A1, compound 1-3, has a Ki value of <0.010 uM.
  • In Vitro
    Aurora B inhibitor 1 also inhibits JAK3 and JAK2 with Kis of <0.25 μM and <0.10 μM, respectively.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    Aurora Kinase
  • Recptor
    Aurora Kinase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    937276-52-3
  • Formula Weight
    529.97
  • Molecular Formula
    C25H26ClF2N7O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    FC1(CN(C1)C2=NC(O[C@@H]3CN(C(=O)C4=C(F)C=CC(Cl)=C4)CC3)=NC(NC5=NNC(C)=C5)=C2)C6CC6
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. FRAYSSE, Damien, et al. AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS. WO2007059299A1.
molnova catalog
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